Andrew J. WilliamsSuda ChakthongDiane GrayRon M. LawrenceTimothy GallagherUniversity of BristolGlaxoSmithKline plc, United KingdomChulabhorn Research InstituteMahidol University2018-07-242018-07-242003-03-20Organic Letters. Vol.5, No.6 (2003), 811-814152370602-s2.0-0141627559https://repository.li.mahidol.ac.th/handle/20.500.14594/20754(Matrix presented) 1,2-Cyclic sulfamidates undergo regiospecific nucleophilic displacement with either methyl thioglycolate or α-amino esters, followed by lactamization (thermal, base-mediated, or cyanide-catalyzed), to give thiomorpholin-3-ones and piperazin-2-ones.Mahidol UniversityBiochemistry, Genetics and Molecular BiologyChemistryArticleSCOPUS10.1021/ol027418h