Publication:
Iodine/TBHP-Promoted One-Pot Deoxygenation and Direct 2-Sulfonylation of Quinoline N-Oxides with Sodium Sulfinates: Facile and Regioselective Synthesis of 2-Sulfonylquinolines

2

Issued Date

2017-01-01

Resource Type

Article

ISSN

10990690
1434193X

DOI

10.1002/ejoc.201601443

Other identifier(s)

2-s2.0-85011969720

Rights

Mahidol University

Rights Holder(s)

SCOPUS

Bibliographic Citation

European Journal of Organic Chemistry. Vol.2017, No.5 (2017), 1025-1032

Suggested Citation

Ladawan Sumunnee, Chonchanok Buathongjan, Chaleena Pimpasri, Sirilata Yotphan Iodine/TBHP-Promoted One-Pot Deoxygenation and Direct 2-Sulfonylation of Quinoline N-Oxides with Sodium Sulfinates: Facile and Regioselective Synthesis of 2-Sulfonylquinolines. European Journal of Organic Chemistry. Vol.2017, No.5 (2017), 1025-1032. doi:10.1002/ejoc.201601443 Retrieved from: https://repository.li.mahidol.ac.th/handle/123456789/42267

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Title

Iodine/TBHP-Promoted One-Pot Deoxygenation and Direct 2-Sulfonylation of Quinoline N-Oxides with Sodium Sulfinates: Facile and Regioselective Synthesis of 2-Sulfonylquinolines

Author(s)

Ladawan Sumunnee
 Chonchanok Buathongjan
 Chaleena Pimpasri
 Sirilata Yotphan

Other Contributor(s)

Mahidol University

Abstract

© 2017 WILEY-VCH Verlag GmbH & Co. KGaA, Weinheim A highly efficient iodine/TBHP-mediated one-pot deoxygenative and regioselective 2-sulfonylation of quinoline N-oxides with sodium sulfinate salts has been developed. This metal-, base-, and phosphorus-free protocol employs readily accessible and easy-to-handle reagents and can be conveniently carried out at room temperature under mild conditions, providing an alternative access to a series of 2-sulfonylquinolines and other related heteroaryl sulfone products in moderate-to-excellent yields within a short reaction time.

Keyword(s)

Chemistry

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URI

https://repository.li.mahidol.ac.th/handle/123456789/42267

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Scopus 2016-2017