Publication: Facile syntheses of 3-halo and mixed 3,5-dihalo analogues of N-acetyl-l-tyrosine via sulfonic acid-catalysed regioselective monohalogenation
dc.contributor.author | Pakorn Bovonsombat | en_US |
dc.contributor.author | Pratheep Khanthapura | en_US |
dc.contributor.author | Michael M. Krause | en_US |
dc.contributor.author | Juthamard Leykajarakul | en_US |
dc.contributor.other | Mahidol University | en_US |
dc.date.accessioned | 2018-07-12T02:16:01Z | |
dc.date.available | 2018-07-12T02:16:01Z | |
dc.date.issued | 2008-12-01 | en_US |
dc.description.abstract | The combination of catalytic amounts of p-toluenesulfonic acid and 1 equiv of N-halosuccinimide afforded highly selective ring-halogenation of N-acetyl-l-tyrosine, furnishing either N-acetyl-3-halo-l-tyrosine analogues or mixed 3,5-dihalo derivatives in a one-pot reaction with excellent yields at room temperature. © 2008 Elsevier Ltd. All rights reserved. | en_US |
dc.identifier.citation | Tetrahedron Letters. Vol.49, No.49 (2008), 7008-7011 | en_US |
dc.identifier.doi | 10.1016/j.tetlet.2008.09.123 | en_US |
dc.identifier.issn | 00404039 | en_US |
dc.identifier.other | 2-s2.0-54049083330 | en_US |
dc.identifier.uri | https://repository.li.mahidol.ac.th/handle/20.500.14594/18807 | |
dc.rights | Mahidol University | en_US |
dc.rights.holder | SCOPUS | en_US |
dc.source.uri | https://www.scopus.com/inward/record.uri?partnerID=HzOxMe3b&scp=54049083330&origin=inward | en_US |
dc.subject | Biochemistry, Genetics and Molecular Biology | en_US |
dc.subject | Chemistry | en_US |
dc.subject | Pharmacology, Toxicology and Pharmaceutics | en_US |
dc.title | Facile syntheses of 3-halo and mixed 3,5-dihalo analogues of N-acetyl-l-tyrosine via sulfonic acid-catalysed regioselective monohalogenation | en_US |
dc.type | Article | en_US |
dspace.entity.type | Publication | |
mu.datasource.scopus | https://www.scopus.com/inward/record.uri?partnerID=HzOxMe3b&scp=54049083330&origin=inward | en_US |